5-HT1A modulator 4

5-HT1A modulator 4 (Compound 1) is a ligand of 5-HT receptors. 5-HT1A modulator 4 has Ki values of 2.18 μM and 19.7 μM for 5-HT1A and 5-HT2A, respectively[1].

Product Specifications

CAS Number

[145208-86-2]

UNSPSC

12352005

Hazard Statement

H302-H315-H319-H335

Target

5-HT Receptor

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Others

Smiles

CN1CCN(C2=NC=CC=N2)CC1

Molecular Formula

C9H14N4

Molecular Weight

178.23

Precautions

P261-P264-P270-P271-P280-P302+P352-P304+P340-P305+P351+P338-P330-P362+P364-P403+P233-P405-P501

References & Citations

[1]Mokrosz MJ, et al. Structure-activity relationship studies of CNS agents, Part 25. 4,6-di (heteroaryl) -2- (N-methylpiperazino) pyrimidines as new, potent 5-HT2A receptor ligands: a verification of the topographic model. Arch Pharm (Weinheim) . 1995 Sep;328 (9) :659-66.