8-Cyclopentyl-1,3-dimethylxanthine (Standard)

8-Cyclopentyl-1,3-dimethylxanthine (Compound 2a) is a selective adenosine A1 receptor antagonist with Kis of 10.9 nM and 1440 nM for A1 receptor and A2 receptor, respectively[1].

Product Specifications

CAS Number

[35873-49-5]

UNSPSC

12352005

Target

Adenosine Receptor

Related Pathways

GPCR/G Protein

Field of Research

Cardiovascular Disease

Smiles

O=C(N1C)N(C)C2=C(N=C(C3CCCC3)N2)C1=O

Molecular Formula

C12H16N4O2

Molecular Weight

248.28

References & Citations

[1]K A Jacobson, et al. Sulfur-containing 1,3-dialkylxanthine derivatives as selective antagonists at A1-adenosine receptors. J Med Chem. 1989 Aug;32 (8) :1873-9.