[Dmt1]DALDA
[Dmt1]DALDA is a potent and long-acting analgesic binds to the mu opioid receptor with high affinity and selectivity. [Dmt1]DALDA is a full agonist at hMOR (Kd = 0.199 nM) and hDOR, but only partial agonist against hKOR[1][2].
Product Specifications
CAS Number
[255861-98-4]
UNSPSC
12352209
Target
Opioid Receptor
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Others
Smiles
CC(C=C(C=C1C)O)=C1C[C@H](N)C(N[C@H](CCCNC(N)=N)C(N[C@H](C(N[C@H](C(N)=O)CCCCN)=O)CC2=CC=CC=C2)=O)=O
Molecular Formula
C32H49N9O5
Molecular Weight
639.79
References & Citations
[1]Zhao, G. M., et al., (2003) . Comparison of [Dmt1]DALDA and DAMGO in binding and G protein activation at mu, delta, and kappa opioid receptors. The Journal of pharmacology and experimental therapeutics, 307 (3), 947–954.
Shipping Conditions
Room temperature
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-P5131/
Scientific Category
Peptides
Clinical Information
No Development Reported
Curated Selection
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