Des-threoninol-octreotide
Des-threoninol-octreotide (Compound 13) is a Somatostatin analog. Des-threoninol-octreotide inhibits cloned somatostatin receptors with IC50 values of 13.62 nM, 10.63 nM, 10.95 nM for mSSTR2b, rSSTR5 and hSSTR5, respectively[1].
Product Specifications
CAS Number
[160841-00-9]
UNSPSC
12352209
Target
Somatostatin Receptor
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Metabolic Disease
Smiles
O=C(N[C@@H](CSSC[C@@H](C(O)=O)NC1=O)C(N[C@@H](CC2=CC=CC=C2)C(N[C@H](CC3=CNC4=CC=CC=C34)C(N[C@@H](CCCCN)C(N[C@H]1[C@H](O)C)=O)=O)=O)=O)[C@@H](CC5=CC=CC=C5)N
Molecular Formula
C45H57N9O9S2
Molecular Weight
932.12
References & Citations
[1]Osapay G, et al. Lanthionine-somatostatin analogs: synthesis, characterization, biological activity, and enzymatic stability studies. J Med Chem. 1997 Jul 4;40 (14) :2241-51.
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
No Development Reported
Curated Selection
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