CTX-1211
CTX-1211 is a selective, orally effective melanocortin MC4R agonist (EC50=0.38 nM). CTX-1211 can enhance the feeding suppression and weight loss effects induced by liraglutide , and promote anorexia and weight loss activity. CTX-1211 is mainly used in the study of obesity and other metabolic disorders[1].
Product Specifications
UNSPSC
12352209
Target
Melanocortin Receptor
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Metabolic Disease
Smiles
O=C(N[C@@H](CCCNC(N)=N)C(N[C@@H](CSSC[C@@H](C(N)=O)NC1=O)C(N[C@@H](CC(O)=O)C(N[C@@H](C)C(N[C@@H](CCCNC(N)=N)C(N[C@@H](CC(O)=O)C(N[C@@H](CC2=CC=CC=C2)C(N[C@@H](CCCNC(N)=N)C(N[C@H]1CC3=CNC4=CC=CC=C34)=O)=O)=O)=O)=O)=O)=O)=O)C
Molecular Formula
C57H83N21O15S2
Molecular Weight
1366.53
References & Citations
[1]Dahir NS, et al. Inhibition of the melanocortin-3 receptor (MC3R) causes generalized sensitization to anorectic agents. bioRxiv [Preprint]. 2023 Dec 7:2023.12.05.570114.
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
No Development Reported
Isoform
MC4R
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
GTR15099912 1 Vial
Lentiviral human TULP4 shRNA (UAS) - Lentiviral human TULP4 shRNA (UAS, RFP) (100)
Sign In for Pricing
View Details 
GTR10403718 96 Well
Human 26S proteasome non ATPase regulatory subunit 13 (PSMD13) ELISA kit
Sign In for Pricing
View Details