Nesiritide (acetate)
Nesiritide (Brain Natriuretic Peptide-32 human) acetate is a recombinant human B-type natriuretic peptide. Nesiritide acetate is a NPRs agonist, with Kd values of 7.3 and 13 pM for NPR-A and NPR-C, respectively. Nesiritide acetate regulates V1/2 activation/inactivation of the L-type calcium channel. Nesiritide acetate shows vasodilatory, diuretic, and natriuretic activities. Nesiritide acetate is used in cardiovascular diseases such as heart failure and vascular remodeling after arterial injury[1][2][3][4][5][6][7].
Product Specifications
Product Name Alternative
Brain Natriuretic Peptide-32 human (acetate) ; BNP-32 (acetate)
UNSPSC
12352209
Target
Calcium Channel; Natriuretic Peptide Receptor (NPR)
Related Pathways
GPCR/G Protein; Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Smiles
Molecular Formula
C145H248N50O44S4
Molecular Weight
3524.09
References & Citations
Shipping Conditions
Room temperature
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-P0003A/
Scientific Category
Peptides
Clinical Information
Phase 4
CAS Number
[1684439-46-0]
Available Sizes
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