(R) -AZ8838
(R) -AZ8838 is a competitive PAR2 antagonist with a pKi of 5.2 for human PAR2. (R) -AZ8838 exert anti-inflammatory effects in a rat model of PAR2 agonist-induced paw oedema[1].
Product Specifications
CAS Number
[2151021-59-7]
UNSPSC
12352005
Target
Protease Activated Receptor (PAR)
Related Pathways
GPCR/G Protein
Field of Research
Inflammation/Immunology
Smiles
O[C@@H](C1=NC=CN1)C2=C(C=C(C=C2)F)CCC
Molecular Formula
C13H15FN2O
Molecular Weight
234.27
References & Citations
[1]Nawwar M A M, et al. Flavonoids of the flowers of Tamarix nilotica[J]. Phytochemistry, 1984, 23 (10) : 2347-2349.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
PAR2
Curated Selection
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