P2Y2R antagonist 1
P2Y2R antagonist 1 is a selective P2Y2R antagonist (pIC50 = 7.78) . P2Y2R antagonist 1 can be used for the study of Glioma[1].
Product Specifications
UNSPSC
12352005
Target
P2Y Receptor
Related Pathways
GPCR/G Protein
Field of Research
Cancer
Smiles
O=C(C1=CC=C(CN(C(N2)=O)C=C(C3C4=CC=C(C)C=C4C=CC5=CC(C)=CC=C35)C2=S)O1)NC6=CC7=C(N(CC)C(CC7)=O)C=C6
Molecular Formula
C38H34N4O4S
Molecular Weight
642.77
References & Citations
[1]Abdalrahman RAM, et al. From tetrazole to isoquinolinone: Structure-based optimization and late-stage diversification of AR-C118925-derived P2Y2 receptor antagonists. Eur J Med Chem. 2026 Jan 15;302 (Pt 2) :118335.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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