E3 Ligase Ligand-linker Conjugate 214
E3 Ligase Ligand-linker Conjugate 214 is an E3 ligase ligand-linker conjugate containing a Von Hippel-Lindau (VHL) ligand and a linker. E3 Ligase Ligand-linker Conjugate 214 can bind to a target protein ligand to form a PROTAC molecule, PROTAC LSD1 Degrader 1 (HY-179229) [1].
Product Specifications
CAS Number
[2451247-91-7]
UNSPSC
12352005
Target
PROTAC-Linker Conjugates for PAC
Related Pathways
Antibody-drug Conjugate/ADC Related; PROTAC
Field of Research
Cancer
Smiles
CC1=C(SC=N1)C2=CC=C(C=C2)CNC([C@@H]3C[C@H](CN3C([C@H](C(C)(C)C)NC(CCCCCCCCCCCN)=O)=O)O)=O
Molecular Formula
C34H53N5O4S
Molecular Weight
627.88
References & Citations
[1]Coulson ME, et al. Synthetic and structure-activity studies of SP2577 and TCP towards LSD1 targeting PROTACs. RSC Med Chem. 2025 Aug 5;16 (10) :4952-4959.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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