(S) -5-HT2CR agonist 1
(S) -5-HT2CR agonist 1 (Compound (S) -16k) is selective 5-HT2CR agonist, with an EC50 of 14 nM. FXa-IN-2 can be used in the research of hyperlocomotion[1].
Product Specifications
CAS Number
2841458-00-0
UNSPSC
12352005
Target
5-HT Receptor
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Neurological Disease
Smiles
OC1=C(C2=C3[C@@]([H])(NCCC3=C1)CC4=C2C(Cl)=CC=C4)OC.Cl
Molecular Formula
C17H17Cl2NO2
Molecular Weight
338.23
References & Citations
[1]Qin W, et al. Discovery of New N-H Aporphine Derivatives As Brain-Penetrant Gq-Biased 5-HT2C Receptor Agonists and Dual 5-HT2C/5-HT2A Receptor Agonists. J Med Chem. 2025 Nov 13;68 (21) :23300-23323.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
5-HT2 Receptor
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