V1b Receptor antagonist-1
V1b receptor antagonist-1 is a potent, selective and brain-penetrant vasopressin 1b (V1b) receptor antagonist. V1b receptor antagonist-1 exhibits anti-depressant activity. V1b receptor antagonist-1 can be used for the research of neurological disease, such as depression[1].
Product Specifications
CAS Number
1056550-56-1
UNSPSC
12352005
Target
Vasopressin Receptor
Related Pathways
GPCR/G Protein
Field of Research
Neurological Disease
Smiles
N#CC1=CC=C2C(C(C3=CC(OC)=CC=C3OCC)(N4CCN(CC4)C5=CC=NC=C5)C(N2S(=O)(C6=CC=CC7=CC=CN=C76)=O)=O)=C1
Molecular Formula
C36H32N6O5S
Molecular Weight
660.74
References & Citations
[1]Geneste H, et al. Novel, potent, selective and brain penetrant vasopressin 1b receptor antagonists. Bioorg Med Chem Lett. 2018 Oct 15;28 (19) :3260-3264.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
V1b Receptor
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