V1b Receptor antagonist-1
V1b receptor antagonist-1 is a potent, selective and brain-penetrant vasopressin 1b (V1b) receptor antagonist. V1b receptor antagonist-1 exhibits anti-depressant activity. V1b receptor antagonist-1 can be used for the research of neurological disease, such as depression[1].
Product Specifications
CAS Number
[1056550-56-1]
UNSPSC
12352005
Target
Vasopressin Receptor
Related Pathways
GPCR/G Protein
Field of Research
Neurological Disease
Smiles
N#CC1=CC=C2C(C(C3=CC(OC)=CC=C3OCC)(N4CCN(CC4)C5=CC=NC=C5)C(N2S(=O)(C6=CC=CC7=CC=CN=C76)=O)=O)=C1
Molecular Formula
C36H32N6O5S
Molecular Weight
660.74
References & Citations
[1]Geneste H, et al. Novel, potent, selective and brain penetrant vasopressin 1b receptor antagonists. Bioorg Med Chem Lett. 2018 Oct 15;28 (19) :3260-3264.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
V1b Receptor
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
