RSK2-IN-6
RSK2-IN-5 (compoud C2) is a p90 ribosomal S6 kinase 2 (RSK2) inhibitor with a Kd of 856 nM. RSK2-IN-5 exhibits antitumor activity against breast cancer and melanoma cancer cells[1].
Product Specifications
CAS Number
304474-86-0
UNSPSC
12352005
Target
Ribosomal S6 Kinase (RSK)
Related Pathways
MAPK/ERK Pathway
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Smiles
O=C(C1=CC=CC([N+]([O-])=O)=C1)NNC2=C3C(CCCC4)=C4SC3=NC=N2
Molecular Formula
C17H15N5O3S
Molecular Weight
369.40
References & Citations
[1]Yue Zhao, et al. Discovery of novel p90 ribosomal S6 kinase 2 inhibitors for potential cancer treatment through ligand-based and structure-based virtual screening methods. Chemometrics and Intelligent Laboratory Systems. Volume 217, 15 October 2021, 104402
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
C0013-32B-PE 200 µL
CBLB, ID (E3 Ubiquitin-protein Ligase CBL-B, Signal Transduction Protein CBL-B, SH3-binding Protein CBL-B, Casitas B-lineage Lymphoma Proto-oncogene b, RING Finger Protein 56, Nbla00127, RNF56) (PE) discontinued
Sign In for Pricing
View Details 
KLB2383 1x 96 Well
GENLISA™ Bovine Platelet Derived Growth Factor Subunit B (PDGFB) ELISA
Sign In for Pricing
View Details 
K2128504 1.0 µg DNA
SETD7 sgRNA CRISPR Lentivector (Human) (Target 3)
Sign In for Pricing
View Details