SST1 receptor antagonist-1
SST1 receptor antagonist-1 (Compound 23) is a selective Somatostatin receptor 1 (SST1) antagonist with pKds of 9.11 and 8.79 for rSST1 and hSST1, respectively. SST1 receptor antagonist-1 can be used for retinal and endocrine dysfunctions, cancer and neuropsychiatric disorders research[1].
Product Specifications
CAS Number
[868057-23-2]
UNSPSC
12352005
Target
Somatostatin Receptor
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Cancer; Endocrinology; Neurological Disease
Smiles
O=C(CCN(CCC1C2=C(OC3=C1C=CC=C3)C=CC=C2)C)N4CCN(CC4)C5=CC=C(C(F)=C5)F
Molecular Formula
C29H31F2N3O2
Molecular Weight
491.57
References & Citations
[1]Troxler T, et al. Discovery of novel non-peptidic beta-alanine piperazine amide derivatives and their optimization to achiral, easily accessible, potent and selective somatostatin sst1 receptor antagonists. Bioorg Med Chem Lett. 2009 Mar 1;19 (5) :1305-9.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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