CDD-1132

CDD-1132 (Compound 8) is a potent inhibitor of BRDT-BD2. CDD-1132 has an IC50 of 13 nM against BRDT-BD2. CDD-1132 can be studied in research on nonhormonal contraceptive agent[1].

Product Specifications

CAS Number

[2757619-83-1]

UNSPSC

12352005

Target

Epigenetic Reader Domain

Related Pathways

Epigenetics

Field of Research

Endocrinology

Smiles

O=C(C1=CC(C(C2=CC3=C(N2C)C=CC=C3)=NN4C)=C4C=C1)NC5=CC=C(C)C(NC(C6=CC=C(C(NC)=O)C=C6)=O)=C5

Molecular Formula

C34H30N6O3

Molecular Weight

570.64

References & Citations

[1]Yu, Z., et al., (2021) . Discovery and characterization of bromodomain 2-specific inhibitors of BRDT. Proceedings of the National Academy of Sciences of the United States of America, 118 (9), e2021102118.