Asuptegravir

Asuptegravir (Compound 1) is an inhibitor of HIV integrase activity. Asuptegravir inhibits HIV in HEK293T cells (EC50 = 1.08 nM) . Asuptegravir can be studied in anti-AIDs/HIV research[1].

Product Specifications

CAS Number

[2765212-92-6]

UNSPSC

12352005

Target

HIV

Related Pathways

Anti-infection

Field of Research

Infection

Smiles

C[C@@H]1C2(CO[C@]3([H])N1C(C(N(C=C4C(NCC5=C(C=C(C=C5)F)F)=O)C3)=C(O)C4=O)=O)CC2

Molecular Formula

C22H21F2N3O5

Molecular Weight

445.42

References & Citations

[1]Yian Shi, et al., Polycyclic carbamoylpyridone derivatives, process for their preparation and pharmaceutical compositions containing them. CN114230579A.