TRPMPZQ-IN-1
TRPMPZQ-IN-1 (Compound 52) is a TRPMPZQ inhibitor, with an EC50 of 0.38 μM against TRPMPZQ from Spirometra erinaceieuropaei. TRPMPZQ-IN-1 exhibits antiparasitic activity, showing an EC50 of 4.3 μM against Echinococcus multilocularis. TRPMPZQ-IN-1 can be used in antiparasitic research[1].
Product Specifications
UNSPSC
12352100
Target
Parasite; TRP Channel
Related Pathways
Anti-infection; Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
COVID-19-immunoregulation
Field of Research
Infection
Smiles
O=C(N1CC(N2CCC3=CC=CC=C3[C@@H]2C1)=S)C4CCSCC4
Molecular Formula
C18H22N2OS2
Molecular Weight
346.51
References & Citations
[1]Sprague DJ, et al. Target-Based Design of Praziquantel Analogs at Cestode TRPMPZQ. ACS Infect Dis. 2025 Aug 3.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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