RXFP1 receptor agonist-9
RXFP1 receptor agonist-9 is a potent RXFP1 agonist with an EC50 of 2.5 μM and Ymax of 65%. RXFP1 receptor agonist-9 exhibits good microsomal stability, reasonable PK and pharmacological activity. RXFP1 receptor agonist-9 can be used to the study of heart failure[1].
Product Specifications
CAS Number
[2924765-23-9]
UNSPSC
12352005
Target
RXFP Receptor
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Smiles
O=C(N[C@@H]1[C@@H]2CC[C@H]([C@@H]1C(NC3=CC(C(F)(F)F)=C(C=C3)F)=O)/C2=C/C4CC4)C5=CC(C6=C(C=CC(C(C(O)=O)OC(NC)=O)=C6)F)=CC=C5OC
Molecular Formula
C37H34F5N3O7
Molecular Weight
727.67
References & Citations
[1]Su S et, al. The Discovery of C7-Substituted Norbornyl Bisamides as RXFP1 Small Molecule Agonists. J Med Chem. 2025 Jun 12;68 (11) :12185-12203.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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