WDR5-MYC-IN-2
WDR5-MYC-IN-2 is an inhibitor of WDR5-MYC protein-protein interaction (PPI) with IC50 of 0.59 μM. WDR5-MYC-IN-2 can be studied in research for MYC-driven cancer and development of other effective WDR5-MYC PPI inhibitors[1].
Product Specifications
CAS Number
[3062125-47-4]
UNSPSC
12352005
Target
C-Myc; WDR5
Related Pathways
Apoptosis; Epigenetics
Field of Research
Cancer
Smiles
BrC1=CC(S(=O)(NC2=CC(C3=CN(C)N=C3)=C(NC(C45CCCC5)=O)C4=C2)=O)=C(O)C(Cl)=C1
Molecular Formula
C22H20BrClN4O4S
Molecular Weight
551.84
References & Citations
[1]Sun, W., et al., (2025) . Discovery of Novel Inhibitors for WD Repeat-Containing Protein 5 (WDR5) -MYC Protein-Protein Interaction. Chemical biology & drug design, 105 (5), e70129.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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