GABAB receptor antagonist 4
GABAB receptor antagonist 4 (Compound 28) is a GABAB receptor antagonist. GABAB receptor antagonist 4 can inhibit GABA-induced G protein activation. GABAB receptor antagonist 4 competitively binds to the orthosteric site of GABAB receptor. GABAB receptor antagonist 4 can be used to study GABAB receptor-related neurological diseases[1].
Product Specifications
CAS Number
[91981-93-0]
UNSPSC
12352005
Target
GABA Receptor
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Field of Research
Neurological Disease
Smiles
CN(C(N=C(N=[N+]=[N-])N1C)=C1C(N2)=O)C2=O
Molecular Formula
C7H7N7O2
Molecular Weight
221.18
References & Citations
[1]Evenseth LSM, et al. Identification of Orthosteric GABAB Receptor Ligands by Virtual Screening and In Vitro Validation. ACS Omega. 2025 May 16;10 (21) :22005-22017.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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