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USP7 activator 1

USP7 activator 1 (compound MS-8) is an activator of USP7 by engaging the allosteric C-terminal binding pocket of USP7[1].

Product Specifications

CAS Number

[868940-26-5]

UNSPSC

12352005

Target

Deubiquitinase

Related Pathways

Cell Cycle/DNA Damage

Applications

Cancer-programmed cell death

Field of Research

Cancer

Purity

99.24

Smiles

O=C(C1(C)N(CCN(C)C)C(C2=CC(OC=C3)=C3N2C1)=O)NC4CCCCCC4

Molecular Formula

C22H32N4O3

Molecular Weight

400.51

References & Citations

[1]Isabella Jaen Maisonet, et al. Small-molecule allosteric activator of ubiquitin-specific protease 7 (USP7) . bioRxiv. 2025 Mar 16:2025.03.14.643379.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

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