BDM_92499
BDM_92499 is a nanomolar selective IRAP inhibitor, with an IC50 of 3.4 nM. BDM_92499 also inhibits ERAP1 and ERAP2, with IC50 values of 0.46 μM and 4.2 μM, respectively[1].
Product Specifications
UNSPSC
12352005
Target
Aminopeptidase
Related Pathways
Metabolic Enzyme/Protease
Field of Research
Others
Smiles
NC([C@@H](NC(C(CC(C)C)C(NO)=O)=O)CC1=CNC2=CC=C(OCC3=CC=CC=C3)C=C21)=O
Molecular Formula
C25H30N4O5
Molecular Weight
466.53
References & Citations
[1]Ben He, et al. Discovery of New Nanomolar Selective IRAP Inhibitors. J Med Chem. 2025 Feb 27;68 (4) :4168-4195.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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