OT-R agonist 1 (TFA)
OT-R agonist 1 TFA (compound 5) is an oxytocin receptor agonist with an EC50 of 0.39 nM. OT-R agonist 1 TFA shows V1A antagonist activity with an EC50 of 2432 nM and can be used for study of CNS disorders[1].
Product Specifications
CAS Number
[3039925-73-7]
UNSPSC
12352005
Target
Oxytocin Receptor; Vasopressin Receptor
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Smiles
FC(F)(F)C(O)=O.CC1=CC(C(N2CC3=C(NC4=CC=CC=C42)N(C)N=C3)=O)=CC=C1CNC(N5C[C@H](OCC6=CC(O)=CC(O)=C6)C[C@H]5C(N(C)C)=S)=O
Molecular Formula
C37H40F3N7O7S
Molecular Weight
783.82
References & Citations
[1]Li Y, et al. Novel Nonpeptide as Oxytocin Receptor Agonist. ACS Med Chem Lett. 2025 Apr 21;16 (5) :750-751.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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