Rocavorexant
Rocavorexant is the antagonist for orexin-1 receptor with pIC50 of 9.1 for human OX1 (while pIC50 for human OX2 is 6.0) [1].
Product Specifications
CAS Number
2115665-09-1
UNSPSC
12352005
Target
Orexin Receptor (OX Receptor)
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Neurological Disease
Smiles
FC(F)(F)C1=CN=C(C=N1)NC[C@H](C)N(C)C(C2=C(N3N=CC=N3)C=CC(C)=N2)=O
Molecular Formula
C18H19F3N8O
Molecular Weight
420.39
References & Citations
[1]Martin B, et al. Therapeutic compounds. WO2017129829
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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