Amezalpat
Amezalpat is the antagonist for PPARα with IC50 of 58 nM. Amezalpat exhibits antineoplastic activity[1].
Product Specifications
CAS Number
[1616372-41-8]
Product Name Alternative
TPST-1120
UNSPSC
12352005
Target
PPAR
Related Pathways
Cell Cycle/DNA Damage; Metabolic Enzyme/Protease; Vitamin D Related/Nuclear Receptor
Applications
Cancer-programmed cell death
Field of Research
Cancer
Purity
99.8500
Smiles
O=C(CC1=CC(C2=CC(CCCC3=NN(CC4=CC=C(C(C)(C)C)C=C4)C(N3CC)=O)=CC=C2)=CC=C1OCC)O
Molecular Formula
C34H41N3O4
Molecular Weight
555.71
References & Citations
[1]Stock NS, et al., Triazolone compounds and uses thereof. WO2014099503.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
PPARα
Available Sizes
Curated Selection
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