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NUAK1-IN-2

NUAK1-IN-2 (Compound 24) is a NUAK1 (IC50 of 3.162 nM) and CDK2/4/6 inhibitor. NUAK1-IN-2 can be used in cancer, neurodevelopmental disorders and Alzheimer's disease research[1].

Product Specifications

UNSPSC

12352005

Target

AMPK; CDK

Related Pathways

Cell Cycle/DNA Damage; Epigenetics; PI3K/Akt/mTOR

Field of Research

Cancer; Neurological Disease

Smiles

CN1C(C2)CC1CN2C(C=C3)=CC=C3NC4=NC5=C(C=CN5CC6CCOCC6)C=N4

Molecular Formula

C24H30N6O

Molecular Weight

418.53

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

CDK2; CDK4; CDK6

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