Lp (a) -IN-5
Lp (a) -IN-5 (Compound A) is an orally active lipoprotein (a) (Lp (a) ) inhibitor. Lp (a) -IN-5 inhibits the assembly of Apo (a) and ApoB proteins with an IC50 value of 0.41 nM. Lp (a) -IN-5 is promising for research of diseases related to elevated plasma Lp (a) levels, such as cardiovascular diseases[1].
Product Specifications
CAS Number
2924841-79-0
UNSPSC
12352211
Target
Apolipoprotein
Related Pathways
Metabolic Enzyme/Protease
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Smiles
O=C(O)[C@H]([C@H]1CCNC1)CC2=CC=CC(CN(CC3=CC(C[C@H](C(O)=O)[C@H]4CCNC4)=CC=C3)CCOC5=CC(C[C@H](C(O)=O)[C@H]6CCNC6)=CC=C5)=C2
Molecular Formula
C43H56N4O7
Molecular Weight
740.93
References & Citations
[1]Yao JQ, et al. Crystal form of lipoprotein compound and preparation method therefor. WO2024230805A1. 2024-11-14.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
Explore Other Products
Browse additional items from our catalog
Titin (TTN, Connectin, Rhabdomyosarcoma Antigen MU-RMS-40.14) (HRP)
