FEKAP
FEKAP is a brain-penetrant and selective kappa opioid receptor (KOR) agonist (Ki = 0.43 nM) which isotope labeled form exhibits excellent imaging properties. 11C-FEKAP can be utilized as a radiotracer for imaging KOR[1].
Product Specifications
CAS Number
[2324155-84-0]
UNSPSC
12352005
Target
Opioid Receptor
Related Pathways
GPCR/G Protein; Neuronal Signaling
Smiles
FCCN(CC)C[C@H]1N(CCN(C1)C(OC)=O)C(CC2=CC(Cl)=C(C=C2)Cl)=O
Molecular Formula
C19H26Cl2FN3O3
Molecular Weight
434.33
References & Citations
[1]Li S, et al. Novel Kappa Opioid Receptor Agonist as Improved PET Radiotracer: Development and in Vivo Evaluation. Mol Pharm. 2019 Apr 1;16 (4) :1523-1531.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
κ Opioid Receptor/KOR
Curated Selection
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