5-HT2A antagonist 3
5-HT2A antagonist 3 (Formula (III) ) is a 5-HT2A receptor antagonist and inverse agonist with a pIC50 of 8.7 and a pKi of 9. 5-HT2A antagonist 3 can be utilized in neurological reesearch[1].
Product Specifications
CAS Number
1134815-69-2
UNSPSC
12352005
Target
5-HT Receptor
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Smiles
O=C(N(C1CCN(CC1)C)CC2=CC=C(C=C2)F)NCC3=CC=C(C=C3)OCC(C)(C)O
Molecular Formula
C25H34FN3O3
Molecular Weight
443.55
References & Citations
[1]Henriette K.U., et al. N-substituted piperidine derivatives as serotonin receptor agents. WO2009039461A2. 2009-03-26
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
5-HT2 Receptor; α-1 microglobulin
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