P5SA-2
P5SA-2 is a selective allosteric activator of PPP5C. P5SA-2 exerts its effects by modulating the phosphatase domain of PPP5C and can increase PPP5C activity by 3.2-fold at 100 μM with an apparent affinity constant of 7.8 μM. P5SA-2 can be used in cancer and Alzheimer's disease research[1].
Product Specifications
CAS Number
864717-20-4
UNSPSC
12352005
Target
Phosphatase
Related Pathways
Metabolic Enzyme/Protease
Field of Research
Cancer; Neurological Disease
Purity
99.51
Smiles
ClC1=CC=C(CC2=NOC(C3=CC(OC)=C(OC)C=C3)=N2)C=C1
Molecular Formula
C17H15ClN2O3
Molecular Weight
330.77
References & Citations
[1]Zhang H, et al. Dual function of protein phosphatase 5 (PPP5C) : An emerging therapeutic target for drug discovery. Eur J Med Chem. 2023 Jun 5;254:115350.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C (Powder, protect from light)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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