NSD2-PWWP1-IN-1
NSD2-PWWP1-IN-1 (compound 31) is a potent NSD2-PWWP1 inhibitor with an IC50 value of 0.64 µM. NSD2-PWWP1-IN-1 has the potential for the research of cancer[1].
Product Specifications
CAS Number
2797183-30-1
UNSPSC
12352005
Target
Histone Methyltransferase
Related Pathways
Epigenetics
Field of Research
Cancer
Purity
98.72
Smiles
N#CC1=C2C=CC=CC2=C(C3=C(C4=C(C)C=C(CNC(C)(C)C)C=C4C)N=CN3C)C=C1
Molecular Formula
C28H30N4
Molecular Weight
422.56
References & Citations
[1]Li N, et al. Structure-Based Discovery of a Series of NSD2-PWWP1 Inhibitors. J Med Chem. 2022 Jul 14;65 (13) :9459-9477.
Shipping Conditions
Room Temperature
Storage Conditions
Store at room temperature, keep dry and cool
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
NSD2/MMSET/WHSC1
Available Sizes
Frequently Asked Questions
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