CDK9 ligand 3
CDK9 ligand 3 is the ligand for CDK9 and can be used for synthesis of PROTAC degrader PROTAC CDK9 degrader-11 (HY-170978) [1].
Product Specifications
CAS Number
[3039540-24-1]
UNSPSC
12352005
Target
CDK; Ligands for Target Protein for PROTAC
Related Pathways
Cell Cycle/DNA Damage; PROTAC
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Smiles
O=C(NC1=CNN=C1C(NC2CCN(CC2)C(CBr)=O)=O)C3=C(C=CC=C3Cl)Cl
Molecular Formula
C18H18BrCl2N5O3
Molecular Weight
503.18
References & Citations
[1]Wang Y, et al., Identification of a Potent and Selective CDK9 Degrader as a Targeted Therapeutic Option for the Treatment of Small-Cell Lung Cancer. J Med Chem. 2025 Feb 13;68 (3) :2528-2550.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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