P2X4 antagonist-3
P2X4 antagonist-3 (Compound 14c) is a P2X4 antagonist with an IC50 value of 1.2 μM. P2X4 antagonist-3 is promising for research of neuroinflammation, chronic pain, and cancer progression[1].
Product Specifications
UNSPSC
12352005
Target
P2X Receptor
Related Pathways
Membrane Transporter/Ion Channel
Field of Research
Cancer; Inflammation/Immunology; Neurological Disease
Smiles
O=C(N1C(COC2=CC=C(OCO3)C3=C2)CNCC1)NC4=CC=C(F)C=C4
Molecular Formula
C19H20FN3O4
Molecular Weight
373.38
References & Citations
[1]Erlitz KS, et al. Piperazine-based P2X4 receptor antagonists. Arch Pharm (Weinheim) . 2025 Jan;358 (1) :e2400860.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
P2X4 Receptor
Curated Selection
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