H1R ligand-1
H1R ligand-1 (Compound fragment 1) is a high-affinity ligand for the human histamine H1 receptor (H1R) . H1R ligand-1 can be used as a scaffold to design and synthesize a set of derivatives to explore H1R binding kinetics[1].
Product Specifications
CAS Number
19642-70-7
UNSPSC
12352005
Target
Histamine Receptor
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling
Field of Research
Neurological Disease
Smiles
CN1CCC(OC2=CC=CC=C2CC3=CC=CC=C3)CC1
Molecular Formula
C19H23NO
Molecular Weight
281.39
References & Citations
[1]Kuhne S, et al. Probing the Histamine H1 Receptor Binding Site to Explore Ligand Binding Kinetics. J Med Chem. 2025 Jan 9;68 (1) :448-464.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
H1 Receptor
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