GRK6-IN-5
GRK6-IN-5 is a GRK6 polypeptide inhibitor, with IC50 value of 4.48 μΜ. GRK6-IN-5 can be used to study hematological malignancies, inflammation diseases, and autoimmune disorders[1].
Product Specifications
CAS Number
[33495-39-5]
UNSPSC
12352005
Target
G Protein-coupled Receptor Kinase (GRK)
Related Pathways
GPCR/G Protein
Field of Research
Cancer; Inflammation/Immunology
Smiles
OC1=C(C(C2=NC=CC=C2)NC3=CC=C(C=C3)OCC)C=CC4=CC=CN=C14
Molecular Formula
C23H21N3O2
Molecular Weight
371.43
References & Citations
[1]Alexander Keith Stewart, et al. Inhibiting g protein coupled receptor 6 kinase polypeptides. WO2013063458. WIPO. 2012-10-26.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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