Anti-inflammatory agent 94

Anti-inflammatory agent 94 (compound 4b) is a potent cannabinoid ligand with Kis of 29 nM and 8 nM against CB2 and CB1. Anti-inflammatory agent 94 can be utilized in inflammation rersearch[1].

Product Specifications

CAS Number

[501927-29-3]

UNSPSC

12352005

Target

Cannabinoid Receptor

Related Pathways

GPCR/G Protein; Neuronal Signaling

Field of Research

Inflammation/Immunology; Neurological Disease

Smiles

C[C@]1(C[C@](CC1)([H])C2(C)C)[C@@H]2NC(C3=C(C)N(C4=C(OC)C=CC=C43)CCN5CCOCC5)=O

Molecular Formula

C27H39N3O3

Molecular Weight

453.62

References & Citations

[1]Wrobleski ST, et al. Rational design and synthesis of an orally active indolopyridone as a novel conformationally constrained cannabinoid ligand possessing antiinflammatory properties. J Med Chem. 2003 May 22;46 (11) :2110-6.