Setipiprant (Standard)
Setipiprant (Standard) is the analytical standard of Setipiprant. This product is intended for research and analytical applications. Setipiprant (ACT-129968) is an orally active and selective CRTH2 antagonist. Setipiprant interacts with hCRTH2 receptor with an IC50 value of 6 nM. Setipiprant inhibits prostanoid receptors hDP1 and hEP2 with IC50 values of 1290 and 2600 nM, respectively. Setipiprant can be used for the research of asthma and rhinitis[1].
Product Specifications
CAS Number
866460-33-5
UNSPSC
12352100
Target
CRTH2 (GPR44) ; Prostaglandin Receptor; Reference Standards
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Others
Field of Research
Inflammation/Immunology; Endocrinology
Smiles
O=C(O)CN1C2=C(CN(C(C3=C4C=CC=CC4=CC=C3)=O)CC2)C5=C1C=CC(F)=C5
Molecular Formula
C24H19FN2O3
Molecular Weight
402.42
References & Citations
Shipping Conditions
Room temperature
Scientific Category
Reference Standards
Available Sizes
Frequently Asked Questions
Explore Other Products
Browse additional items from our catalog
LMX1B (LIM homeobox Transcription Factor 1-beta, LIM/homeobox Protein 1.2, LMX-1.2, LIM/homeobox Protein LMX1B, LMX1B) discontinued
LMX1B (LIM homeobox Transcription Factor 1-beta, LIM/homeobox Protein 1.2, LMX-1.2, LIM/homeobox Protein LMX1B, LMX1B) discontinued
Rabbit anti-human karyopherin (importin) beta 1 polyclonal Antibody