Emupertinib
Emupertinib (example 37) is a potent EGFR inhibitor with IC50 values of [1].
Product Specifications
CAS Number
[2472802-77-8]
UNSPSC
12352005
Target
EGFR
Related Pathways
JAK/STAT Signaling; Protein Tyrosine Kinase/RTK
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Smiles
O=C(C1=NC=C(C)N=C1)NC23CCC(CC2)(C3)N4C(C#C)=C(C5=C4N=CN=C5N)C6=CC7=C(C=CC=C7)N=C6
Molecular Formula
C30H26N8O
Molecular Weight
514.58
References & Citations
[1] , et al. 7H-pyrrolo [2,3-d] pyrimidine-4-amine derivative.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
EGFR/ErbB1/HER1
Curated Selection
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