Gabapentin enacarbil (Standard)
Gabapentin enacarbil (Standard) is the analytical standard of Gabapentin enacarbil. This product is intended for research and analytical applications. Gabapentin enacarbil (XP-13512) is a prodrug of Gabapentin designed to be absorbed throughout the intestine by high-capacity nutrient transporters. Gabapentin is a potent, orally active P/Q type Ca2+ channel blocker. Gabapentin enacarbil can be used for the study of Restless Legs Syndrome (RLS) and postherpetic neuralgia (PHN)[2].
Product Specifications
CAS Number
478296-72-9
UNSPSC
12352100
Target
Calcium Channel; Reference Standards
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling; Others
Field of Research
Neurological Disease
Smiles
O=C(O)CC1(CNC(OC(OC(C(C)C)=O)C)=O)CCCCC1
Molecular Formula
C16H27NO6
Molecular Weight
329.39
References & Citations
[1]Cundy KC, et al. XP13512 [ (+/-) -1- ([ (alpha-isobutanoyloxyethoxy) carbonyl] aminomethyl) -1-cyclohexane acetic acid], a novel gabapentin prodrug: I. Design, synthesis, enzymatic conversion to gabapentin, and transport by intestinal solute transporters. J Pharmacol Exp Ther. 2004 Oct;311 (1) :315-23.|[2]Cundy KC, et al. XP13512 [ (+/-) -1- ([ (alpha-isobutanoyloxyethoxy) carbonyl] aminomethyl) -1-cyclohexane acetic acid], a novel gabapentin prodrug: II. Improved oral bioavailability, dose proportionality, and colonic absorption compared with gabapentin in rats and monkeys. J Pharmacol Exp Ther. 2004 Oct;311 (1) :324-33.
Shipping Conditions
Room temperature
Scientific Category
Reference Standards
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