Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

Entospletinib (Standard)

Entospletinib (Standard) is the analytical standard of Entospletinib. This product is intended for research and analytical applications. Entospletinib (GS-9973) is an orally bioavailable, selective Syk inhibitor with an IC50 of 7.7 nM.

Product Specifications

CAS Number

1229208-44-9

UNSPSC

12352100

Target

Reference Standards; Syk

Related Pathways

Others; Protein Tyrosine Kinase/RTK

Field of Research

Cancer

Smiles

C12=NC=CN1C=C(C3=CC4=C(C=C3)C=NN4)N=C2NC5=CC=C(N6CCOCC6)C=C5

Molecular Formula

C23H21N7O

Molecular Weight

411.46

References & Citations

[1]Currie KS, et al. Discovery of GS-9973, a Selective and Orally Efficacious Inhibitor of Spleen Tyrosine Kinase. J Med Chem. 2014 May 8;57 (9) :3856-73.|[2]Burke RT, et al. A potential therapeutic strategy for chronic lymphocytic leukemia by combining Idelalisib and GS-9973, a novel spleen tyrosine kinase (Syk) inhibitor. Oncotarget. 2014 Feb 28;5 (4) :908-15.

Shipping Conditions

Room temperature

Scientific Category

Reference Standards

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

TEM1 (CD248) Mouse Monoclonal Antibody (Biotin conjugated) [Clone ID: OTI1H6]
TA807065AM 100 µL

TEM1 (CD248) Mouse Monoclonal Antibody (Biotin conjugated) [Clone ID: OTI1H6]

Sign In for Pricing
View Details
PRPF38B Human Gene Knockout Kit (CRISPR)
KN423346 1 Kit

PRPF38B Human Gene Knockout Kit (CRISPR)

Sign In for Pricing
View Details
Recombinant gamma Catenin Antibody
RC-16940-01 50 μL

Recombinant gamma Catenin Antibody

Sign In for Pricing
View Details
Recombinant gamma Catenin Antibody
RC-16940-02 100 µL

Recombinant gamma Catenin Antibody

Sign In for Pricing
View Details
Recombinant gamma Catenin Antibody
RC-16940-03 1 mL

Recombinant gamma Catenin Antibody

Sign In for Pricing
View Details
2-Chloro-4’-hydroxybenzophenone
TRC-C366690-250MG 250 mg

2-Chloro-4’-hydroxybenzophenone

Sign In for Pricing
View Details