Revefenacin-d4
Revefenacin-d4 (TD-4208-d4) is deuterium labeled Revefenacin. Revefenacin (TD-4208; GSK1160724) is a potent mAChR antagonist; has a high affinity on M3 receptor with a Ki of 0.18 nM.
Product Specifications
Product Name Alternative
TD-4208-d4; GSK1160724-d4
UNSPSC
12352005
Target
Isotope-Labeled Compounds
Related Pathways
Others
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology; Cardiovascular Disease
Smiles
O=C(NC1=CC=CC=C1C2=CC=CC=C2)OC3CCN(CC3)CCN(C)C(C4=C(C([2H])=C(C([2H])=C4[2H])CN5CCC(CC5)C(N)=O)[2H])=O
Molecular Formula
C35H39D4N5O4
Molecular Weight
601.77
References & Citations
[1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53 (2) :211-216.
Shipping Conditions
Room temperature
Scientific Category
Isotope-Labeled Compounds
Clinical Information
No Development Reported
Curated Selection
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