Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

Cav 3.1 blocker 1

Cav 3.1 blocker 1 (compound 12) is a T-type calcium channel blocker with an IC50value of 160 nM for Cav3.1. Cav 3.1 blocker 1 weakly inhibits Cav 3.2 (IC50 of 5000 nM), and shows no inhibition on Cav 3.3 and Cav 1.2 (IC50 of >10000 nM) [1].

Product Specifications

CAS Number

2158201-04-6

UNSPSC

12352005

Target

Calcium Channel

Related Pathways

Membrane Transporter/Ion Channel; Neuronal Signaling

Field of Research

Neurological Disease

Smiles

O=C(C1=NN(C(C2=CC=CC=C2)=C1C(F)F)C3=CC=C(C=C3)F)NCC4=C(OCC(F)(F)F)C=CC=C4

Molecular Formula

C26H19F6N3O2

Molecular Weight

519.44

References & Citations

[1]Bezençon O, et al. Milestones to the Discovery of T-type Calcium Channel Blockers for the Treatment of Generalized Epilepsies. Chimia (Aarau) . 2017 Oct 25;71 (10) :722-729.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

T-type calcium channel

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Recombinant Human CAVEOLIN2/CAV2 protein (GST, His tag)
PDEH100962-01 20 µg

Recombinant Human CAVEOLIN2/CAV2 protein (GST, His tag)

Sign In for Pricing
View Details
Recombinant Human CAVEOLIN2/CAV2 protein (GST, His tag)
PDEH100962-02 100 µg

Recombinant Human CAVEOLIN2/CAV2 protein (GST, His tag)

Sign In for Pricing
View Details
Recombinant Human CAVEOLIN2/CAV2 protein (GST, His tag)
PDEH100962-03 500 µg

Recombinant Human CAVEOLIN2/CAV2 protein (GST, His tag)

Sign In for Pricing
View Details
Recombinant Human CAVEOLIN2/CAV2 protein (GST, His tag)
PDEH100962-04 1 mg

Recombinant Human CAVEOLIN2/CAV2 protein (GST, His tag)

Sign In for Pricing
View Details
SIAH Interacting Protein (CACYBP) Mouse Monoclonal Antibody [Clone ID: AT3G8]
AM50340PU-N 100 µL

SIAH Interacting Protein (CACYBP) Mouse Monoclonal Antibody [Clone ID: AT3G8]

Sign In for Pricing
View Details
Elab Fluor® Red 780 Anti-Mouse CD48 Antibody[HM48-1]
E-AB-F1017S-01 50 Tests

Elab Fluor® Red 780 Anti-Mouse CD48 Antibody[HM48-1]

Sign In for Pricing
View Details