Telmapitant
Telmapitant is an orally active NK1R antagonist. Telmapitant has antiemetic effect and can be used for the research of delayed onset emesis[1].
Product Specifications
CAS Number
[552292-58-7]
UNSPSC
12352005
Target
Neurokinin Receptor
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Others
Smiles
O=C(N1)N[C@]2(CN[C@@](C3=CC=CC=C3)(CO[C@@H](C4=CC(C(F)(F)F)=CC(C(F)(F)F)=C4)C)CC2)C1=O
Molecular Formula
C24H23F6N3O3
Molecular Weight
515.45
References & Citations
[1]Chen-Chao Wang, et al. Oral pharmaceutical composition of an nk-1 antagonist. WO2019122068A1. 2020-06-21
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
NK1R
Curated Selection
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