DS39201083

DS39201083, a Conolidine derivative, is a potent and orally active analgesic agent. DS39201083 shows no agonist activity at the mu opioid receptor. DS39201083 can be used for the study of neurological diseases[1].

Product Specifications

CAS Number

[2361560-81-6]

UNSPSC

12352005

Target

Opioid Receptor

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Smiles

O=C1C2=C(CN3CCC1(CC3)C)C4=C(C=CC=C4)N2

Molecular Formula

C16H18N2O

Molecular Weight

254.33

References & Citations

[1]Arita T, et al. Discovery of conolidine derivative DS39201083 as a potent novel analgesic without mu opioid agonist activity. Bioorg Med Chem Lett. 2019 Aug 1;29 (15) :1938-1942.