GRK6-IN-4

GRK6-IN-4 is a G protein coupled receptor 6 kinase (GRK6) inhibitor with an IC50 of 1.56 μM. GRK6-IN-4 can be utilized in research related to hematological malignancies, inflammatory diseases, and autoimmune disorders[1].

Product Specifications

CAS Number

[300731-73-1]

UNSPSC

12352005

Hazard Statement

H315-H319-H320

Target

G Protein-coupled Receptor Kinase (GRK)

Related Pathways

GPCR/G Protein

Field of Research

Cancer; Inflammation/Immunology

Smiles

N#CC1=C(N)N(CCCC)C2=C1N=C3C=CC=CC3=N2

Molecular Formula

C15H15N5

Molecular Weight

265.31

Precautions

P264-P280-P302+P352-P305+P351+P338-P362

References & Citations

[1]Alexander K.S., et al. Inhibiting g protein coupled receptor 6 kinase polypeptides. WO2013063458A2. 2013-05-02

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

Phase 1

Curated Selection

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