BMS-830216
BMS-830216 is an antagonist of MCHR-1. BMS-830216 is a phosphate ester prodrug. BMS-830216 can be studied in obesity-related research[1].
Product Specifications
CAS Number
[1197420-06-6]
UNSPSC
12352005
Target
MCHR1 (GPR24)
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Smiles
ClC1=CC=C(C2=CC(N=CN(C3=CC(OC)=C(OC[C@H](OP(O)(O)=O)C4CC4)C=C3)C5=O)=C5S2)C=C1
Molecular Formula
C24H22ClN2O7PS
Molecular Weight
548.93
References & Citations
[1]Washburn, W. N., et al., (2014) . Identification of a nonbasic melanin hormone receptor 1 antagonist as an antiobesity clinical candidate. Journal of medicinal chemistry, 57 (18), 7509-7522.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 1
Curated Selection
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