Contilisant
Contilisant is a permeable antioxidant and neuroprotectant agent. Contilisant exhibits high nM affinity at H3R. Contilisant inhibits monoamine oxidases and cholinesterases. Contilisant has a binding affinity of 65.23 nM towards hS1R. Contilisant can significantly restore cognitive deficit induced by Aβ1-42 in the radial maze assay of Alzheimer’s animal model[1].
Product Specifications
CAS Number
2135615-68-6
UNSPSC
12352005
Target
Cholinesterase (ChE) ; Histamine Receptor; Monoamine Oxidase; Reactive Oxygen Species (ROS)
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Metabolic Enzyme/Protease; Neuronal Signaling; NF-κB
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease; Neurological Disease
Smiles
C#CCN(C)CC(N1C)=CC2=C1C=CC(OCCCN3CCCCC3)=C2
Molecular Formula
C22H31N3O
Molecular Weight
353.50
References & Citations
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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