GR-175737
GR 175737 is a partial histamine H3 receptor agonist, with an EC50 of 7.8 nM. GR 175737 can be used in the research of inflammatory diseases[1].
Product Specifications
CAS Number
176860-26-7
UNSPSC
12352005
Target
Histamine Receptor
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling
Field of Research
Inflammation/Immunology
Smiles
ClC1=CC=C(C=C1)CC2=NOC(CCC3=CN=CN3)=N2
Molecular Formula
C14H13ClN4O
Molecular Weight
288.73
References & Citations
[1]Soudijn W, et al. Structure–activity relationships of inverse agonists for G‐protein‐coupled receptors. Medicinal research reviews, 2005, 25 (4) : 398-426.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
H3 Receptor
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