L-796778 (acetate)
L-796778 acetate is a selective agonist of the sst3 receptor. In CHO-K1 cells expressing the hsst3 receptor, L-796778 acetate is a partial agonist that inhibits Forskolin -stimulated cAMP production with an IC50 value of 18 nM. L-796778 acetate has anticonvulsant effect[1].
Product Specifications
CAS Number
2922280-21-3
UNSPSC
12352211
Target
Somatostatin Receptor
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Purity
98.00
Smiles
O=C([C@H](CCCCN)NC([C@@H](CCCC)NC(N[C@H](C(NC1=CC=C(C=C1)[N+]([O-])=O)=O)CC2=CC=CC=C2)=O)=O)OC.CC(O)=O
Molecular Formula
C31H44N6O9
Molecular Weight
644.72
References & Citations
[1]Pfeiffer M, et al. Homo- and heterodimerization of somatostatin receptor subtypes. Inactivation of sst (3) receptor function by heterodimerization with sst (2A) . J Biol Chem. 2001 Apr 27;276 (17) :14027-36.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C (Powder, stored under nitrogen, away from moisture)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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