P2Y1 antagonist 1
P2Y1 antagonist 1 (compound 10q) is a potent antagonist of P2Y1, with the IC50s of 1.1 nM and 0.24 μM in FLIPR assay and hPA assay, respectively. P2Y1 antagonist 1 plays an important role in antiplatelet research[1].
Product Specifications
CAS Number
1555697-67-0
UNSPSC
12352005
Target
P2Y Receptor
Related Pathways
GPCR/G Protein
Field of Research
Cardiovascular Disease
Smiles
O=C(NC1=CC=C(OC(F)(F)F)C=C1)NC2=CC=CC=C2N3CC(C)(C)C4=C3C(O)=CC(F)=C4C5=CC=C(Cl)C=C5
Molecular Formula
C30H24ClF4N3O3
Molecular Weight
585.98
References & Citations
[1]Wu Yang, et al. Discovery of 4‑Aryl-7-Hydroxyindoline-Based P2Y1 Antagonists as Novel Antiplatelet Agents. J Med Chem. 2014 Jul 24;57 (14) :6150-64.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
P2Y1 Receptor
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