P2Y1 antagonist 1
P2Y1 antagonist 1 (compound 10q) is a potent antagonist of P2Y1, with the IC50s of 1.1 nM and 0.24 μM in FLIPR assay and hPA assay, respectively. P2Y1 antagonist 1 plays an important role in antiplatelet research[1].
Product Specifications
CAS Number
1555697-67-0
UNSPSC
12352005
Target
P2Y Receptor
Related Pathways
GPCR/G Protein
Field of Research
Cardiovascular Disease
Smiles
O=C(NC1=CC=C(OC(F)(F)F)C=C1)NC2=CC=CC=C2N3CC(C)(C)C4=C3C(O)=CC(F)=C4C5=CC=C(Cl)C=C5
Molecular Formula
C30H24ClF4N3O3
Molecular Weight
585.98
References & Citations
[1]Wu Yang, et al. Discovery of 4‑Aryl-7-Hydroxyindoline-Based P2Y1 Antagonists as Novel Antiplatelet Agents. J Med Chem. 2014 Jul 24;57 (14) :6150-64.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
P2Y1 Receptor
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
BNC680034-500 1x 500 µL
Cytokeratin 8/18 (C-51), CF568 conjugate, 0.1mg/mL
Sign In for Pricing
View Details 
BNC940630-100 1x 100 µL
Mucin 1 / EMA / Episialin / CD227 (VU-2G7), CF594 conjugate, 0.1mg/mL
Sign In for Pricing
View Details 
BNC040948-100 1x 100 µL
Cytokeratin 5/8 (C-50), CF405S conjugate, 0.1mg/mL
Sign In for Pricing
View Details 
BNC682038-100 1x 100 µL
Gp100 / Melanosome / PMEL17 / SILV (Melanoma Marker) (PMEL/2038), CF568 conjugate, 0.1mg/mL
Sign In for Pricing
View Details 
BNC741991-500 1x 500 µL
Cytokeratin 20 (KRT20) (Colorectal Epithelial Marker) (KRT20/1991), CF740 conjugate, 0.1mg/mL
Sign In for Pricing
View Details